Basic Peptide Information

DICL ID
DICL_Pep_00281
Ion Channel
Neuronal acetylcholine receptor subunit alpha-9/alpha-10
Peptide Function
Inhibitor
Gene Name
Chrna9/Chrna10

Activity Data (nM)

IC50
4.61 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
TCRSSGRYCRSPYDRRRRYCRRITDACV
Peptide UniProt Accession
UniParc
UPI00085DE742
Peptide Synonyms/Alias
[CHEMBL4553407; GeXIVA[1;4]; GLXC-27609; BDBM50520487; TC(1)RSSGRYC(2)RSPYDRRRRYC(2)RRITDAC(1)V; Thr-Cys(1)-Arg-Ser-Ser-Gly-Arg-Tyr-Cys(2)-Arg-Ser-Pro-Tyr-Asp-Arg-Arg-Arg-Arg-Tyr-Cys(2)-Arg-Arg-Ile-Thr-Asp-Ala-Cys(1)-Val]
Peptide Species
Conus generalis (General cone)
Peptide Name
Alpha-conotoxin GeXIVA
CAS Number
Not available

Experimental Conditions

pH
pH 9.6
Holding Potential (mV)
Not specified
Temperature
25 ± 1 °C
Test Method
Binding assay
Test Species
Not specified

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available